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  5. Tocris Bioscience™ Selpercatinib

Tocris Bioscience™ Selpercatinib
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Código de producto. 18759196
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Cantidad:
10 mg
50 mg
Tamaño de la unidad:
10 miligramos
50 miligramos
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Código de producto. Cantidad unitSize
18759196 50 mg 50 miligramos
18747026 10 mg 10 miligramos
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Código de producto. 18759196 Proveedor Tocris Bioscience™ N.º de proveedor 7696/50

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Descripción

Potent and selective RET inhibitor

Selpercatinib, is a potent and selective receptor tyrosine kinase RET inhibitor (EC50 = 4 nM). It shows > 100-fold selectivity for > 95% of 228 purified kinase domains in radiometric assays. In vitro, it inhibits proliferation of cancer cell lines containing RET mutations or gene fusions. In vivo, it inhibits tumor growth in diverse RET mouse models. Selpercatinib is orally bioavailable.
TRUSTED_SUSTAINABILITY

Especificaciones

Nombre del producto químico o material 6-(2-Hydroxy-2-methylpropoxy)-4-[6-[6-[(6-methoxy-3-pyridinyl)methyl]-3,6-diazabicyclo[3.1.1 ]hept-3-yl]-3-pyridinyl]pyrazolo[1,5-a]pyridine-3-carbonitrile
CAS 2152628-33-4
Cantidad 50 mg
Objetivo Ret
Fórmula molecular C29H31N7O3
Pureza 0.98
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